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| Product Name | AKR1C3 Inhibitor I |
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| Description | Purity >98% by HPLC. A highly potent and selective inhibitor of the type 5 17-Beta-hydroxysteroid dehydrogenase AKR1C3. In repeat assays it showed an IC50 of 0.013 ± 0.003 MM for AKR1C3, compared with 20.3 ± 3.8 MM against AKR1C1 and >30 MM against AKR1C2 and AKR1C4. This inhibitor also showed potency in a cellular assay, blocking the ability of AKR1C3 to metabolize a proven substrate. Does not display any COX (cyclooxygenase) inhibition at 10 µM in whole blood assay. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 3-(3,4-Dihydroisoquinolin2(1H)-ylsulfonyl)benzoic acid |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | LS-H2977 |
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| Order / More Info | AKR1C3 Inhibitor I from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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