| 产品详情 |
| Edit |   |
|---|
| Product Name | Amiselimod (hydrochloride) |
|---|
| Description | Purity >95%. Amiselimod is a prodrug that is converted to (S)-amiselimod phosphate by sphingosine kinases. Amiselimod phosphate is a highly selective S1P1 receptor antagonist (EC50 = 74 pM) that is without activity at S1P3 receptors. It is approximately five-fold weaker as an activator of G protein-coupled inwardly rectifying K+ (GIRK) channels than fingolimod phosphate. Amiselimod is orally bioavailable and has minimal cardiac effects when tested clinically. |
|---|
| Size | n/a |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | 2-amino-2-[2-[4-(heptyloxy)-3-(trifluoromethyl)phenyl]ethyl]-1,3-propanediol, monohydrochloride, MT-1303 |
|---|
| Gene, Accession, CAS # | CAS: 942398-84-7 |
|---|
| Catalog # | LS-H6514 |
|---|
| Price | |
|---|
| Order / More Info | Amiselimod (hydrochloride) from LIFESPAN BIOSCIENCES INC. |
|---|
| Product Specific References | n/a |
|---|
| 产品资料 |
|
|