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| Product Name | NVS-CECR2-1 |
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| Description | Purity >95%. NVS-CECR2-1 is a potent inhibitor of CECR2 (cat eye syndrome chromosome region, candidate 2), a component of chromatin complexes that regulate gene expression controlling development. It binds CECR2 with high affinity (IC50 = 0.047 µM by Alpha screen, Kd = 0.80 µM by ITC). NVS-CECR2-1 demonstrates no crossreactivity in a panel of 48 bromodomains and has no major activity in kinase, protease, and receptor panels. It shows robust activity in cells by FRAP assay, due to its slow off-rate, and has no acute toxicity. See the Structural Genomics Consortium (SGC) website for more information. |
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| Size | n/a |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-cyclopropyl-2-(propylsulfonyl)-6-[1-(2,2,6,6-tetramethyl-4-piperidinyl)-1H-indol-5-yl]-4-pyrimidinamine, NVS-1 |
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| Gene, Accession, CAS # | CAS: 1992047-61-6 |
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| Catalog # | LS-H9119 |
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| Order / More Info | NVS-CECR2-1 from LIFESPAN BIOSCIENCES INC. |
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| Product Specific References | n/a |
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