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| Product Name | UBP 310 |
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| Description | GluK1 (formerly GLUK5) kainate receptor antagonist (IC50 = 130 nM); also blocks recombinant homomeric GluK3 (forrmerly GLUK7) receptors. Displays 12,700-fold selectivity for GluK1 (formerly GLUK5) over GluK2 (formerly GLUK6). Exhibits no activity at mGlu group I or NMDA receptors at concentrations of up to 10 μM. Apparent KD value is 18 ± 4 nM for depression of kainate responses on the dorsal root. Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions. Purity 98%. MW (observed): 353.35 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-thiophene-3-yl-methyl)-5-methylpyrimidine-2,4-dione |
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| Gene, Accession, CAS # | CAS: 902464-46-4 |
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| Catalog # | 3621/10 |
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| Price | |
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| Order / More Info | UBP 310 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 22205648, 24801624 |
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| 产品资料 |
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