| 产品详情 |
| Edit |   |
| Product Name | MLN2480 |
| Description | Purity >98%. MLN2480 is an orally bioavailable pan-Raf kinase inhibitor that inhibits MAP kinase pathway signaling in BRAF-mutant melanoma models. It shows antitumor activity in melanoma, colon, lung, and pancreatic cancer xenograft models. MLN2480 demonstrates synergistic activity with TAK-733, an allosteric MEK kinase inhibitor. |
| Size | n/a |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 6-amino-5-chloro-N-[(1R)-1-[5-[[[5-chloro-4-(trifluoromethyl)-2-pyridinyl]amino]carbonyl]-2-thiazolyl]ethyl]-4-pyrimidinecarboxamide, BIIB-024, TAK-580 |
| Gene, Accession, CAS # | CAS: 1096708-71-2 |
| Catalog # | LS-H8768 |
| Price | |
| Order / More Info | MLN2480 from LIFESPAN BIOSCIENCES INC. |
| Product Specific References | n/a |
| 产品资料 |
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